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LY 2979165

CAS No. 311385-35-9

LY 2979165( MP-101 | LY2979165 )

Catalog No. M13996 CAS No. 311385-35-9

LY2979165 (MP-101) is the alanine prodrug of LY2812223, a selective orthosteric mGlu2 receptor agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    LY 2979165
  • Note
    Research use only, not for human use.
  • Brief Description
    LY2979165 (MP-101) is the alanine prodrug of LY2812223, a selective orthosteric mGlu2 receptor agonist.
  • Description
    LY2979165 (MP-101) is the alanine prodrug of LY2812223, a selective orthosteric mGlu2 receptor agonist; suppresses glutamate release at presynaptic receptors during periods of enhanced, abnormal, glutamate activity and has potential for use in treating psychiatric and neurologic disorders. Alzheimer Disease Phase 2 Clinical.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MP-101 | LY2979165
  • Pathway
    GPCR/G Protein
  • Target
    mGluR
  • Recptor
    mGluR
  • Research Area
    Neurological Disease
  • Indication
    Alzheimer Disease

Chemical Information

  • CAS Number
    311385-35-9
  • Formula Weight
    355.369
  • Molecular Formula
    C13H17N5O5S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    (1R,2S,4R,5R,6R)-4-((4H-1,2,4-triazol-3-yl)thio)-2-((S)-2-aminopropanamido)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. McColm J, et al. Br J Clin Pharmacol. 2017 Aug;83(8):1654-1667.
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